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原料药&中间体


原料药 API's (Active Pharmaceutical Ingredient's)

免疫抑制剂类
环孢菌素 A, Cyclosporin A 59865-13-3 环孢菌素 H, Cyclosporin H 83602-39-5
环孢菌素 D, Cyclosporin D 63775-96-2 雷帕霉素, Sirolimus (Rapamycin) 53123-88-9
环孢菌素 C, Cyclosporin C 59787-61-0 他克莫司, Tacrolimus (FK506) 104987-11-3
麦考酚酸, Mycophenolic acid 24280-93-1 麦考酚酸酯, Mycophenolate mofetil [115007-34-6] 128794-94-5
抗帕金森
普拉克索, Pramipexole dihydrochloride 104632-26-0 罗匹尼罗, Ropinirole hydrochloride 91374-21-9
抗病毒和抗艾滋
替诺褔韦, Tenofovir disoproxil fumarate 202138-50-9 恩曲他滨, Emtricitabine 143491-57-0
抗癌药
甲磺酸伊马替尼, Imatinib mesylate 220127-57-1 伊马替尼碱, Imatinib base 152459-95-5
马来酸舒尼替尼, Sunitinib malate 341031-54-7 舒尼替尼碱, Sunitinib base 152459-95-5
琥珀酸瓦他拉尼, Vatalanib succinate 212142-18-2 瓦他拉尼碱, Vatalanib base 212141-54-3
盐酸埃罗替尼, Erlotinib hydrochloride 183319-69-9 埃罗替尼碱, Erlotinib base 183321-74-6
二甲苯磺酸拉帕替尼, Lapatinib Ditosylate 388082-78-8 拉帕替尼碱, Lapatinib base 231277-92-2
吉非替尼, Gefitinib 184475-35-2 尼罗替尼, Nilotinib 641571-10-0
喹喏酮类抗菌药
左旋氧氟沙星半水物, Levofloxacin hemihydrate 100986-85-4 盐酸洛美沙星, Lomefloxacin hydrochloride 98079-51-7
其他原料药
氢溴酸槟榔碱, Arecoline hydrobromide 300-08-3 盐酸度洛西汀, Duloxetine hydrochloride 136434-34-9
盐酸丙美卡因, Proxymetacaine hydrochloride 5875-06-9 齐留通, Zileuton 111406-87-2
氟阿尼酮 Fluanisone 1480-19-9 美海屈林萘二磺酸盐, Mebhydrolin napadisylate 6153-33-9
饲料添加剂及兽药
盐酸莱克多巴胺, Ractopamine hydrochloride 90274-24-1 盐酸齐帕特罗, Zilpaterol hydrohloride 119520-06-8
布帕伐醌, Buparvaquone 88426-33-9    

None of the products will be supplied to countries in which this could be in conflict with the existing patents. However the final responsibility lies with the Buyer. 这些产品将不供应任何有专利保护的地区和国家,由此引起的法律责任及一切后果将由采购方承担。


中间体 Intermediates

甲磺酸伊马替尼 Imatinib mesylate [220127-57-1]
4-[(4-Methyl-1-piperazinyl)methyl]benzoic acid dihydrochloride hemihydrate
Cas number: 106261-49-8
N-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine
Cas number: 152460-10-1
N-(5-Nitro-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine
Cas number: 152460-09-8
2-Dimethylamino-1-(3-pyridyl)-2-propene-1-one
Cas: 55314-16-4
2-Methyl-5-nitro phenyl guanidine nitrate
Cas number: 152460-08-7, (152460-07-6 for free base)

马来酸舒尼替尼 Sunitinib Malate [341031-54-7]
5-Formyl-2,4-dimethyl-1H-pyrrole-3-carboxylic acid [253870-02-9]
5-Fluoro-1,3-dihydro-indol-2-one [56341-41-4]

瓦他拉尼 Vatalanib [212141-54-3]
1-chloro-4-(4-pyridylmethyl)phthalazine [101094-85-3]
906531-30-4 for HCl salt, 906531-29-1 for DiHCl salt

埃罗替尼 Erlotinib [183319-69-9]
6,7-bis-(2-Methoxyethoxy)-quinazolin-4(3h)-one [179688-29-0]
4-Chloro-6,7-(2-methoxyethoxy)-quinazoline [183322-18-1]

尼罗替尼 Nilotinib [641571-10-0]
3-[(Aminoiminomethyl)amino]-4-methyl-benzoic acid ethyl ester mononitrate
4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid ethyl ester
4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid

拉帕替尼 Lapatinib [231277-92-2]
[3-Chloro-4-(3-fluorobenzyloxy)-phenyl]-(6-iodoquinazolin-4-yl)-amine

普拉克索 Pramipexole dihydrochloride [104632-26-0]

2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole [106006-83-1]
(6S)-(-)-2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole [106092-09-5]

罗匹尼罗 Ropinirole hydrochloride [91374-21-9]
2-Methyl-3-nitrophenylacetic acid [23876-15-5]
N,N-Dipropyl-2-methyl-3-nitrophenylethanamine [91374-23-1]

Tenofovir disoproxil fumarate [104632-26-0]
Tenofovir, PMPA monohydrate [206184-49-8]
(R)-9-(2-hydroxypropyl) adenine [14047-28-0]
DESMP [31618-90-3]

阿札那韦 Atazanavir[198904-31-3]
BOC-L-Phenylalanine; BOC-L-Phenylalanine methyl ester [13734-34-4]
(2R,3S)-N-Boc-3-Amino-1,2-epoxy-4-phenylbutane [98760-08-8]

利托那韦 Ritonavir [155213-67-5]
2-Isopropyl-4-(methylaminomethyl)thiazole [154212-60-9]
N-(4-nitrophenyloxy-carbonyl)-L-valine methyl ester [106261-49-8]

伐昔洛韦 Valaciclovi [124832-26-4]
CBZ-L-Valine [1149-26-4]

丙美卡因 Proxymetacaine hydrochloride [5875-06-9]
3-Nitro-4-propoxybenzoic acid [35288-44-9]